Palladium-Catalyzed One-Pot Approach to 3-Diarylmethyleneoxindoles from Propiolamidoaryl TriflateReportar como inadecuado




Palladium-Catalyzed One-Pot Approach to 3-Diarylmethyleneoxindoles from Propiolamidoaryl Triflate - Descarga este documento en PDF. Documentación en PDF para descargar gratis. Disponible también para leer online.

Integrated Research Institute of Pharmaceutical Sciences, College of Pharmacy, The Catholic University of Korea, Bucheon-si, Gyeonggi-do 420-743, Korea



These authors contributed equally to this work.





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Academic Editor: Roman Dembinski

Abstract 3-Diarylmethyleneoxindoles have been synthesized from propiolamidoaryl triflate utilizing a palladium-catalyzed one-pot reaction consisting of three successive reactions: Sonogashira, Heck, and Suzuki-Miyaura. This method allows for the production of a complex skeleton of 3-diarylmethyleneoxindole from propiolamidoaryl triflate using a commercially available aryl iodide and arylboronic acid in a simple and efficient way with moderate yield and stereoselectivity. View Full-Text

Keywords: 3-Diarylmethyleneoxindole; one-pot reaction; aryl triflate; palladium-catalyzed reaction 3-Diarylmethyleneoxindole; one-pot reaction; aryl triflate; palladium-catalyzed reaction





Autor: Dahye Lee †, Sunhwa Park †, Yoseb Yu, Kye Jung Shin and Jae Hong Seo *

Fuente: http://mdpi.com/



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